Synthesis and Structure-Activity Relationships of New 2-Phenoxybenzamides with Antiplasmodial Activity
The 2-phenoxybenzamide <b>1</b> from the Medicines for Malaria Venture Malaria Box Project has shown promising multi-stage activity against different strains of <i>P. falciparum</i>. It was successfully synthesized via a retrosynthetic approach. Subsequently, twenty-one new d...
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Autores principales: | Theresa Hermann, Patrick Hochegger, Johanna Dolensky, Werner Seebacher, Eva-Maria Pferschy-Wenzig, Robert Saf, Marcel Kaiser, Pascal Mäser, Robert Weis |
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Formato: | article |
Lenguaje: | EN |
Publicado: |
MDPI AG
2021
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Materias: | |
Acceso en línea: | https://doaj.org/article/176a80a80aa24a23946632a02a7cfb4b |
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