A Rational Design of α-Helix-Shaped Peptides Employing the Hydrogen-Bond Surrogate Approach: A Modulation Strategy for Ras-RasGRF1 Interaction in Neuropsychiatric Disorders

In the last two decades, abnormal Ras (rat sarcoma protein)–ERK (extracellular signal-regulated kinase) signalling in the brain has been involved in a variety of neuropsychiatric disorders, including drug addiction, certain forms of intellectual disability, and autism spectrum disorder. Modulation o...

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Détails bibliographiques
Auteurs principaux: Maria Rita Gulotta, Riccardo Brambilla, Ugo Perricone, Andrea Brancale
Format: article
Langue:EN
Publié: MDPI AG 2021
Sujets:
Ras
R
Accès en ligne:https://doaj.org/article/4557875779384e07be7552d6eaf77b9a
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