A Facile Approach to Bis(isoxazoles), Promising Ligands of the AMPA Receptor

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A Facile Approach to Bis(isoxazoles), Promising Ligands of the AMPA Receptor

A convenient synthetic approach to novel functionalized bis(isoxazoles), the promising bivalent ligands of the AMPA receptor, was elaborated. It was based on the heterocyclization reactions of readily available electrophilic alkenes with the tetranitromethane-triethylamine complex. The structural di...

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Détails bibliographiques
Auteurs principaux:	Dmitry A. Vasilenko, Kirill S. Sadovnikov, Kseniya N. Sedenkova, Dmitry S. Karlov, Eugene V. Radchenko, Yuri K. Grishin, Victor B. Rybakov, Tamara S. Kuznetsova, Vladimir L. Zamoyski, Vladimir V. Grigoriev, Vladimir A. Palyulin, Elena B. Averina
Format:	article
Langue:	EN
Publié:	MDPI AG 2021
Sujets:	heterocycles medicinal chemistry heterocyclization tetranitromethane isoxazole bivalent ligand Organic chemistry QD241-441
Accès en ligne:	https://doaj.org/article/732b363d7e634168a92b75b3ea43dab0
Tags:	Ajouter un tag Pas de tags, Soyez le premier à ajouter un tag!

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