Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones

A series of 2-hetaryl- and 2-(hetaryl)ylidene substituted 5-fluoro-8-nitro-1,3-benzothiazin-4-ones was synthesized by interaction of 2,6-difluoro-3-nitrobenzoylisothiocyanate with C-nucleophiles. Cyclocondensation of polyfluorobenzoylchlorides with aryl and hetaryl thioamides represents new approach...

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Autores principales:	Emiliya V. Nosova, Olga A. Batanova, Nataliya N. Mochulskaya, Galina N. Lipunova
Formato:	article
Lenguaje:	EN RU
Publicado:	Uralʹskij federalʹnyj universitet imeni pervogo Prezidenta Rossii B.N. Elʹcina 2020
Materias:	1,3-benzothiazin-4-ones 2-fluorobenzoylchloride 2-fluorobenzoyl-isothiocyanate indole pyrrole cyanomethylbenzimidazole benzoylmethylbenzimidazole thioamide cyclocondensation tuberculostatics Chemistry QD1-999
Acceso en línea:	https://doaj.org/article/a2182820d5e7436b95e934b59c909682
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spelling	oai:doaj.org-article:a2182820d5e7436b95e934b59c9096822021-12-01T05:53:10ZSynthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones2411-141410.15826/chimtech.2020.7.3.01https://doaj.org/article/a2182820d5e7436b95e934b59c9096822020-09-01T00:00:00Zhttps://journals.urfu.ru/index.php/chimtech/article/view/4537https://doaj.org/toc/2411-1414A series of 2-hetaryl- and 2-(hetaryl)ylidene substituted 5-fluoro-8-nitro-1,3-benzothiazin-4-ones was synthesized by interaction of 2,6-difluoro-3-nitrobenzoylisothiocyanate with C-nucleophiles. Cyclocondensation of polyfluorobenzoylchlorides with aryl and hetaryl thioamides represents new approach to 1,3-benzothiazin-4-ones. Some compounds proved to be promising for further development of tuberculostatic agents.Emiliya V. NosovaOlga A. BatanovaNataliya N. MochulskayaGalina N. LipunovaUralʹskij federalʹnyj universitet imeni pervogo Prezidenta Rossii B.N. Elʹcina article1,3-benzothiazin-4-ones2-fluorobenzoylchloride2-fluorobenzoyl-isothiocyanateindolepyrrolecyanomethylbenzimidazolebenzoylmethylbenzimidazolethioamidecyclocondensationtuberculostaticsChemistryQD1-999ENRUChimica Techno Acta, Vol 7, Iss 3, Pp 96-103 (2020)
institution	DOAJ
collection	DOAJ
language	EN RU
topic	1,3-benzothiazin-4-ones 2-fluorobenzoylchloride 2-fluorobenzoyl-isothiocyanate indole pyrrole cyanomethylbenzimidazole benzoylmethylbenzimidazole thioamide cyclocondensation tuberculostatics Chemistry QD1-999
spellingShingle	1,3-benzothiazin-4-ones 2-fluorobenzoylchloride 2-fluorobenzoyl-isothiocyanate indole pyrrole cyanomethylbenzimidazole benzoylmethylbenzimidazole thioamide cyclocondensation tuberculostatics Chemistry QD1-999 Emiliya V. Nosova Olga A. Batanova Nataliya N. Mochulskaya Galina N. Lipunova Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones
description	A series of 2-hetaryl- and 2-(hetaryl)ylidene substituted 5-fluoro-8-nitro-1,3-benzothiazin-4-ones was synthesized by interaction of 2,6-difluoro-3-nitrobenzoylisothiocyanate with C-nucleophiles. Cyclocondensation of polyfluorobenzoylchlorides with aryl and hetaryl thioamides represents new approach to 1,3-benzothiazin-4-ones. Some compounds proved to be promising for further development of tuberculostatic agents.
format	article
author	Emiliya V. Nosova Olga A. Batanova Nataliya N. Mochulskaya Galina N. Lipunova
author_facet	Emiliya V. Nosova Olga A. Batanova Nataliya N. Mochulskaya Galina N. Lipunova
author_sort	Emiliya V. Nosova
title	Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones
title_short	Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones
title_full	Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones
title_fullStr	Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones
title_full_unstemmed	Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones
title_sort	synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones
publisher	Uralʹskij federalʹnyj universitet imeni pervogo Prezidenta Rossii B.N. Elʹcina
publishDate	2020
url	https://doaj.org/article/a2182820d5e7436b95e934b59c909682
work_keys_str_mv	AT emiliyavnosova syntheticapproachesto2arylhetaryland2hetarylylidenederivativesoffluorinated13benzothiazin4ones AT olgaabatanova syntheticapproachesto2arylhetaryland2hetarylylidenederivativesoffluorinated13benzothiazin4ones AT nataliyanmochulskaya syntheticapproachesto2arylhetaryland2hetarylylidenederivativesoffluorinated13benzothiazin4ones AT galinanlipunova syntheticapproachesto2arylhetaryland2hetarylylidenederivativesoffluorinated13benzothiazin4ones
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Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones

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