The synthesis, antimicrobial activity and docking studies of 6-(1H-benzimidazol-2-yl)-5-methylthieno[2,3-d]pyrimidin-4(3H)-ones with acetamide and 1,2,4-oxadiazol-5-ylmethyl substituents
Aim. To synthesize, study the antimicrobial activity and suggest antimicrobial activity mechanism for the novel derivatives of 6-(1H-benzimidazol-2-yl)-5-methylthieno[2,3-d]pyrimidin-4(3H)-one. Results and discussion. As the result of the targeted modification of 6-(1H-benzimidazol-2-yl)-5-methylth...
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Autores principales: | Sergiy V. Vlasov, Oleksandr V. Borysov, Hanna I. Severina, Sergiy M. Kovalenko, Tetiana P. Osolodchenko, Vitaliy S. Vlasov, Victoriya A. Georgiyants |
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Formato: | article |
Lenguaje: | EN RU UK |
Publicado: |
National University of Pharmacy (Kharkiv, Ukraine)
2021
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Materias: | |
Acceso en línea: | https://doi.org/10.24959/ophcj.21.240775 https://doaj.org/article/c248549c64f247df8e09fe7bbe25133d |
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