Structural determinants and regulation of spontaneous activity in GABAA receptors
GABAA receptors (GABAARs) cause inhibition in the brain by functioning as heteropentamers formed from multiple subunit types. Here, the authors demonstrate that receptors incorporating β3 subunits can spontaneously gate, which is modulated by protein kinases and neurosteroids to affect tonic inhibit...
Enregistré dans:
Auteurs principaux: | Craig A. Sexton, Reka Penzinger, Martin Mortensen, Damian P. Bright, Trevor G. Smart |
---|---|
Format: | article |
Langue: | EN |
Publié: |
Nature Portfolio
2021
|
Sujets: | |
Accès en ligne: | https://doaj.org/article/d345dc169b86449ab9fb68e8dd692c86 |
Tags: |
Ajouter un tag
Pas de tags, Soyez le premier à ajouter un tag!
|
Documents similaires
-
Physiological role for GABAA receptor desensitization in the induction of long-term potentiation at inhibitory synapses
par: Martin Field, et autres
Publié: (2021) -
Structural basis of neurosteroid anesthetic action on GABAA receptors
par: Qiang Chen, et autres
Publié: (2018) -
Characterization of zebrafish GABAA receptor subunits
par: Kenichiro Sadamitsu, et autres
Publié: (2021) -
Regulation of action potential waveforms by axonal GABAA receptors in cortical pyramidal neurons.
par: Yang Xia, et autres
Publié: (2014) -
Structural basis of GABARAP-mediated GABAA receptor trafficking and functions on GABAergic synaptic transmission
par: Jin Ye, et autres
Publié: (2021)