Cross Pharmacological, Biochemical and Computational Studies of a Human Kv3.1b Inhibitor from <i>Androctonus australis</i> Venom

The voltage-gated K<sup>+</sup> channels Kv3.1 display fast activation and deactivation kinetics and are known to have a crucial contribution to the fast-spiking phenotype of certain neurons. AahG50, as a natural product extracted from <i>Androctonus australis hector</i> veno...

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Auteurs principaux: Sonia Maatoug, Amani Cheikh, Oussema Khamessi, Hager Tabka, Zied Landoulsi, Jean-Marie Guigonis, Sylvie Diochot, Saïd Bendahhou, Rym Benkhalifa
Format: article
Langue:EN
Publié: MDPI AG 2021
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Accès en ligne:https://doaj.org/article/f1589d1d72c34914a1494d435f104141
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